TRPC5
|
|
|
Hs |
Activator |
- |
- |
- |
1x10-4 |
|
|
⤷ |
Conc range: 1x10-4 M
|
TRPP2
|
|
|
Hs |
Channel blocker |
- |
- |
- |
1x10-4 |
3 |
|
⤷ |
Conc range: 1x10-4 M
[3]
Voltage:
-50.0 mV
|
TRPC1
|
|
|
Hs |
Channel blocker |
Antagonist |
- |
- |
2x10-5 |
10 |
|
⤷ |
Conc range: 2x10-5 M
[10]
Voltage:
-70.0 mV
|
TRPC3
|
|
|
Hs |
Channel blocker |
Antagonist |
7.0 |
pEC50 |
- |
5 |
|
⤷ |
pEC50
7.0
(EC50 1x10-7 M)
[5]
Voltage:
-60.0 mV
|
TRPA1
|
|
|
Mm |
Channel blocker |
Antagonist |
7.0 |
pIC50 |
- |
8 |
|
⤷ |
pIC50
7.0
[8]
Voltage:
-80.0 mV
|
TRPC6
|
|
|
Mm |
Channel blocker |
Antagonist |
5.7 |
pIC50 |
- |
6 |
|
⤷ |
pIC50
5.7
(IC50 1.9x10-6 M)
[6]
Voltage:
-60.0 mV
|
Navi2.1
|
|
|
Hs |
Channel blocker |
- |
5.6 |
pIC50 |
- |
|
|
⤷ |
pIC50
5.6
(IC50 1.4x10-6 M)
|
TRPML3
|
|
|
Mm |
Channel blocker |
Antagonist |
4.7 |
pIC50 |
- |
9 |
|
⤷ |
pIC50
4.7
(IC50 2x10-5 M)
[9]
Voltage:
-80.0 mV
|
ASIC3
|
|
|
Hs |
Channel blocker |
- |
4.4 |
pIC50 |
- |
1 |
|
⤷ |
pIC50
4.4
(IC50 4x10-5 M)
[1]
|
TRPM3
|
|
|
Hs |
Channel blocker |
Antagonist |
4.0 |
pIC50 |
- |
4,7 |
|
⤷ |
pIC50
4.0
[4,7]
|
TRPV4
|
|
|
Hs |
Channel blocker |
- |
- |
- |
- |
|
|
⤷ |
|
Maxi Cl-
|
|
|
Hs |
Channel blocker (extracellular Gd3+) |
- |
- |
- |
- |
|
|
⤷ |
|