cipargamin [Ligand Id: 9721] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1082723 (Kae609, NITD-609, KAE609, KAE-609, NITD609, Cipargamin)
  • A2A receptor/Adenosine A2a receptor in Human [ChEMBL: CHEMBL251] [GtoPdb: 19] [UniProtKB: P29274]
  • This target only has 0 pki data point
1 CHEMBL1082723_lig_chart_1 Adenosine A2a receptor Human
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  • A3 receptor/Adenosine A3 receptor in Human [ChEMBL: CHEMBL256] [GtoPdb: 21] [UniProtKB: P0DMS8]
  • This target only has 0 pki data point
2 CHEMBL1082723_lig_chart_2 Adenosine A3 receptor Human
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  • α1A-adrenoceptor/Alpha-1a adrenergic receptor in Human [ChEMBL: CHEMBL229] [GtoPdb: 22] [UniProtKB: P35348]
  • This target only has 0 pki data point
3 CHEMBL1082723_lig_chart_3 Alpha-1a adrenergic receptor Human
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  • α2A-adrenoceptor/Alpha-2a adrenergic receptor in Human [ChEMBL: CHEMBL1867] [GtoPdb: 25] [UniProtKB: P08913]
  • This target only has 0 pki data point
4 CHEMBL1082723_lig_chart_4 Alpha-2a adrenergic receptor Human
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  • α2B-adrenoceptor/Alpha-2b adrenergic receptor in Human [ChEMBL: CHEMBL1942] [GtoPdb: 26] [UniProtKB: P18089]
  • This target only has 0 pki data point
5 CHEMBL1082723_lig_chart_5 Alpha-2b adrenergic receptor Human
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  • α2C-adrenoceptor/Alpha-2c adrenergic receptor in Human [ChEMBL: CHEMBL1916] [GtoPdb: 27] [UniProtKB: P18825]
  • This target only has 0 pki data point
6 CHEMBL1082723_lig_chart_6 Alpha-2c adrenergic receptor Human
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  • Androgen receptor/Androgen Receptor in Human [ChEMBL: CHEMBL1871] [GtoPdb: 628] [UniProtKB: P10275]
  • This target only has 0 pki data point
7 CHEMBL1082723_lig_chart_7 Androgen Receptor Human
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  • β1-adrenoceptor/Beta-1 adrenergic receptor in Human [ChEMBL: CHEMBL213] [GtoPdb: 28] [UniProtKB: P08588]
  • This target only has 0 pki data point
8 CHEMBL1082723_lig_chart_8 Beta-1 adrenergic receptor Human
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  • β2-adrenoceptor/Beta-2 adrenergic receptor in Human [ChEMBL: CHEMBL210] [GtoPdb: 29] [UniProtKB: P07550]
  • This target only has 0 pki data point
9 CHEMBL1082723_lig_chart_9 Beta-2 adrenergic receptor Human
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  • β3-adrenoceptor/Beta-3 adrenergic receptor in Human [ChEMBL: CHEMBL246] [GtoPdb: 30] [UniProtKB: P13945]
  • This target only has 0 pki data point
10 CHEMBL1082723_lig_chart_10 Beta-3 adrenergic receptor Human
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  • B1 receptor/Bradykinin B1 receptor in Human [ChEMBL: CHEMBL4308] [GtoPdb: 41] [UniProtKB: P46663]
  • This target only has 0 pki data point
11 CHEMBL1082723_lig_chart_11 Bradykinin B1 receptor Human
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  • B2 receptor/Bradykinin B2 receptor in Human [ChEMBL: CHEMBL3157] [GtoPdb: 42] [UniProtKB: P30411]
  • This target only has 0 pki data point
12 CHEMBL1082723_lig_chart_12 Bradykinin B2 receptor Human
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  • CB1 receptor/Cannabinoid CB1 receptor in Human [ChEMBL: CHEMBL218] [GtoPdb: 56] [UniProtKB: P21554]
  • This target only has 0 pki data point
13 CHEMBL1082723_lig_chart_13 Cannabinoid CB1 receptor Human
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  • CCK1 receptor/Cholecystokinin A receptor in Human [ChEMBL: CHEMBL1901] [GtoPdb: 76] [UniProtKB: P32238]
  • This target only has 0 pki data point
14 CHEMBL1082723_lig_chart_14 Cholecystokinin A receptor Human
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  • CCK2 receptor/Cholecystokinin B receptor in Human [ChEMBL: CHEMBL298] [GtoPdb: 77] [UniProtKB: P32239]
  • This target only has 0 pki data point
15 CHEMBL1082723_lig_chart_15 Cholecystokinin B receptor Human
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  • CRF1 receptor/Corticotropin releasing factor receptor 1 in Human [ChEMBL: CHEMBL1800] [GtoPdb: 212] [UniProtKB: P34998]
  • This target only has 0 pki data point
16 CHEMBL1082723_lig_chart_16 Corticotropin releasing factor receptor 1 Human
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  • CRF2 receptor/Corticotropin releasing factor receptor 2 in Human [ChEMBL: CHEMBL4069] [GtoPdb: 213] [UniProtKB: Q13324]
  • This target only has 0 pki data point
17 CHEMBL1082723_lig_chart_17 Corticotropin releasing factor receptor 2 Human
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  • COX-1 /Cyclooxygenase-1 in Human [ChEMBL: CHEMBL221] [GtoPdb: 1375] [UniProtKB: P23219]
  • This target only has 0 pki data point
18 CHEMBL1082723_lig_chart_18 Cyclooxygenase-1 Human
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  • COX-2 /Cyclooxygenase-2 in Human [ChEMBL: CHEMBL230] [GtoPdb: 1376] [UniProtKB: P35354]
  • This target only has 0 pki data point
19 CHEMBL1082723_lig_chart_19 Cyclooxygenase-2 Human
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  • δ receptor/Delta opioid receptor in Human [ChEMBL: CHEMBL236] [GtoPdb: 317] [UniProtKB: P41143]
  • This target only has 0 pki data point
20 CHEMBL1082723_lig_chart_20 Delta opioid receptor Human
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  • D1 receptor/Dopamine D1 receptor in Human [ChEMBL: CHEMBL2056] [GtoPdb: 214] [UniProtKB: P21728]
  • This target only has 0 pki data point
21 CHEMBL1082723_lig_chart_21 Dopamine D1 receptor Human
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  • D2 receptor/Dopamine D2 receptor in Human [ChEMBL: CHEMBL217] [GtoPdb: 215] [UniProtKB: P14416]
  • This target only has 0 pki data point
22 CHEMBL1082723_lig_chart_22 Dopamine D2 receptor Human
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  • D3 receptor/Dopamine D3 receptor in Human [ChEMBL: CHEMBL234] [GtoPdb: 216] [UniProtKB: P35462]
  • This target only has 0 pki data point
23 CHEMBL1082723_lig_chart_23 Dopamine D3 receptor Human
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  • D4 receptor/Dopamine D4 receptor in Human [ChEMBL: CHEMBL219] [GtoPdb: 217] [UniProtKB: P21917]
  • This target only has 0 pki data point
24 CHEMBL1082723_lig_chart_24 Dopamine D4 receptor Human
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  • DAT/Dopamine transporter in Human [ChEMBL: CHEMBL238] [GtoPdb: 927] [UniProtKB: Q01959]
  • This target only has 0 pki data point
25 CHEMBL1082723_lig_chart_25 Dopamine transporter Human
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  • ETA receptor/Endothelin receptor ET-A in Human [ChEMBL: CHEMBL252] [GtoPdb: 219] [UniProtKB: P25101]
  • This target only has 0 pki data point
26 CHEMBL1082723_lig_chart_26 Endothelin receptor ET-A Human
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  • ETB receptor/Endothelin receptor ET-B in Human [ChEMBL: CHEMBL1785] [GtoPdb: 220] [UniProtKB: P24530]
  • This target only has 0 pki data point
27 CHEMBL1082723_lig_chart_27 Endothelin receptor ET-B Human
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  • Estrogen receptor-α/Estrogen receptor alpha in Human [ChEMBL: CHEMBL206] [GtoPdb: 620] [UniProtKB: P03372]
  • This target only has 0 pki data point
28 CHEMBL1082723_lig_chart_28 Estrogen receptor alpha Human
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  • Estrogen receptor-β/Estrogen receptor beta in Human [ChEMBL: CHEMBL242] [GtoPdb: 621] [UniProtKB: Q92731]
  • This target only has 0 pki data point
29 CHEMBL1082723_lig_chart_29 Estrogen receptor beta Human
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  • GABAA receptor α1 subunit/GABAA receptor β1 subunit/GABAA receptor β3 subunit/GABAA receptor α5 subunit/GABAA receptor α3 subunit/GABAA receptor α2 subunit/GABAA receptor β2 subunit/GABAA receptor α4 subunit/GABAA receptor α6 subunit/GABA-A receptor; agonist GABA site in Human [ChEMBL: CHEMBL2109244] [GtoPdb: 404410412408406405411407409] [UniProtKB: P14867P18505P28472P31644P34903P47869P47870P48169Q16445]
  • This target only has 0 pki data point
30 CHEMBL1082723_lig_chart_30 GABA-A receptor; agonist GABA site Human
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  • GIP receptor/Gastric inhibitory polypeptide receptor in Rat [ChEMBL: CHEMBL5001] [GtoPdb: 248] [UniProtKB: P43219]
  • This target only has 0 pki data point
31 CHEMBL1082723_lig_chart_31 Gastric inhibitory polypeptide receptor Rat
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  • ghrelin receptor/Ghrelin receptor in Human [ChEMBL: CHEMBL4616] [GtoPdb: 246] [UniProtKB: Q92847]
  • This target only has 0 pki data point
32 CHEMBL1082723_lig_chart_32 Ghrelin receptor Human
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  • glucagon receptor/Glucagon receptor in Human [ChEMBL: CHEMBL1985] [GtoPdb: 251] [UniProtKB: P47871]
  • This target only has 0 pki data point
33 CHEMBL1082723_lig_chart_33 Glucagon receptor Human
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  • Glucocorticoid receptor in Human [ChEMBL: CHEMBL2034] [GtoPdb: 625] [UniProtKB: P04150]
  • This target only has 0 pki data point
34 CHEMBL1082723_lig_chart_34 Glucocorticoid receptor Human
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35 CHEMBL1082723_lig_chart_35 Glutamate [NMDA] receptor Human
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  • Kv11.1/HERG in Human [ChEMBL: CHEMBL240] [GtoPdb: 572] [UniProtKB: Q12809]
  • This target only has 0 pki data point
36 CHEMBL1082723_lig_chart_36 HERG Human
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  • H1 receptor/Histamine H1 receptor in Human [ChEMBL: CHEMBL231] [GtoPdb: 262] [UniProtKB: P35367]
  • This target only has 0 pki data point
37 CHEMBL1082723_lig_chart_37 Histamine H1 receptor Human
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  • H2 receptor/Histamine H2 receptor in Human [ChEMBL: CHEMBL1941] [GtoPdb: 263] [UniProtKB: P25021]
  • This target only has 0 pki data point
38 CHEMBL1082723_lig_chart_38 Histamine H2 receptor Human
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  • H3 receptor/Histamine H3 receptor in Human [ChEMBL: CHEMBL264] [GtoPdb: 264] [UniProtKB: Q9Y5N1]
  • This target only has 0 pki data point
39 CHEMBL1082723_lig_chart_39 Histamine H3 receptor Human
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  • HCA2 receptor/Hydroxycarboxylic acid receptor 2 in Human [ChEMBL: CHEMBL3785] [GtoPdb: 312] [UniProtKB: Q8TDS4]
  • This target only has 0 pki data point
40 CHEMBL1082723_lig_chart_40 Hydroxycarboxylic acid receptor 2 Human
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  • κ receptor/Kappa opioid receptor in Human [ChEMBL: CHEMBL237] [GtoPdb: 318] [UniProtKB: P41145]
  • This target only has 0 pki data point
41 CHEMBL1082723_lig_chart_41 Kappa opioid receptor Human
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  • MC3 receptor/Melanocortin receptor 3 in Human [ChEMBL: CHEMBL4644] [GtoPdb: 284] [UniProtKB: P41968]
  • This target only has 0 pki data point
42 CHEMBL1082723_lig_chart_42 Melanocortin receptor 3 Human
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  • MC4 receptor/Melanocortin receptor 4 in Human [ChEMBL: CHEMBL259] [GtoPdb: 285] [UniProtKB: P32245]
  • This target only has 0 pki data point
43 CHEMBL1082723_lig_chart_43 Melanocortin receptor 4 Human
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  • Monoamine oxidase A in Human [ChEMBL: CHEMBL1951] [GtoPdb: 2489] [UniProtKB: P21397]
  • This target only has 0 pki data point
44 CHEMBL1082723_lig_chart_44 Monoamine oxidase A Human
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  • motilin receptor/Motilin receptor in Human [ChEMBL: CHEMBL2203] [GtoPdb: 297] [UniProtKB: O43193]
  • This target only has 0 pki data point
45 CHEMBL1082723_lig_chart_45 Motilin receptor Human
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  • μ receptor/Mu opioid receptor in Human [ChEMBL: CHEMBL233] [GtoPdb: 319] [UniProtKB: P35372]
  • This target only has 0 pki data point
46 CHEMBL1082723_lig_chart_46 Mu opioid receptor Human
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  • M1 receptor/Muscarinic acetylcholine receptor M1 in Human [ChEMBL: CHEMBL216] [GtoPdb: 13] [UniProtKB: P11229]
  • This target only has 0 pki data point
47 CHEMBL1082723_lig_chart_47 Muscarinic acetylcholine receptor M1 Human
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  • M2 receptor/Muscarinic acetylcholine receptor M2 in Human [ChEMBL: CHEMBL211] [GtoPdb: 14] [UniProtKB: P08172]
  • This target only has 0 pki data point
48 CHEMBL1082723_lig_chart_48 Muscarinic acetylcholine receptor M2 Human
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  • M3 receptor/Muscarinic acetylcholine receptor M3 in Human [ChEMBL: CHEMBL245] [GtoPdb: 15] [UniProtKB: P20309]
  • This target only has 0 pki data point
49 CHEMBL1082723_lig_chart_49 Muscarinic acetylcholine receptor M3 Human
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  • NK1 receptor/Neurokinin 1 receptor in Human [ChEMBL: CHEMBL249] [GtoPdb: 360] [UniProtKB: P25103]
  • This target only has 0 pki data point
50 CHEMBL1082723_lig_chart_50 Neurokinin 1 receptor Human
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  • Y1 receptor/Neuropeptide Y receptor type 1 in Human [ChEMBL: CHEMBL4777] [GtoPdb: 305] [UniProtKB: P25929]
  • This target only has 0 pki data point
51 CHEMBL1082723_lig_chart_51 Neuropeptide Y receptor type 1 Human
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  • Y2 receptor/Neuropeptide Y receptor type 2 in Human [ChEMBL: CHEMBL4018] [GtoPdb: 306] [UniProtKB: P49146]
  • This target only has 0 pki data point
52 CHEMBL1082723_lig_chart_52 Neuropeptide Y receptor type 2 Human
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  • NTS1 receptor/Neurotensin receptor 1 in Human [ChEMBL: CHEMBL4123] [GtoPdb: 309] [UniProtKB: P30989]
  • This target only has 0 pki data point
53 CHEMBL1082723_lig_chart_53 Neurotensin receptor 1 Human
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  • NET/Norepinephrine transporter in Human [ChEMBL: CHEMBL222] [GtoPdb: 926] [UniProtKB: P23975]
  • This target only has 0 pki data point
54 CHEMBL1082723_lig_chart_54 Norepinephrine transporter Human
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  • phosphodiesterase 4D/Phosphodiesterase 4D in Human [ChEMBL: CHEMBL288] [GtoPdb: 1303] [UniProtKB: Q08499]
  • This target only has 0 pki data point
55 CHEMBL1082723_lig_chart_55 Phosphodiesterase 4D Human
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  • Plasmodium falciparum [ChEMBL: CHEMBL364]
  • This target only has 0 pki data point
56 CHEMBL1082723_lig_chart_56 Plasmodium falciparum Plasmodium falciparum
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  • Plasmodium falciparum 3D7 [ChEMBL: CHEMBL2366922]
  • This target only has 0 pki data point
57 CHEMBL1082723_lig_chart_57 Plasmodium falciparum 3D7 Plasmodium falciparum 3D7
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  • Plasmodium falciparum (isolate K1 / Thailand) in Plasmodium falciparum K1 [ChEMBL: CHEMBL612856]
  • This target only has 0 pki data point
58 CHEMBL1082723_lig_chart_58 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1
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