|
|
|
α1A-adrenoceptor
|
|
|
Rn |
Antagonist |
Antagonist |
9.5 – 10.2 |
pKi |
- |
6,11 |
|
⤷ |
pKi
9.5 – 10.2
[6,11]
|
α1A-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
9.0 – 9.8 |
pKi |
- |
2-3,5,8-9 |
|
⤷ |
pKi
9.0 – 9.8
[2-3,5,8-9]
|
α1D-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.6 – 9.6 |
pKi |
- |
5,8-9 |
|
⤷ |
pKi
8.6 – 9.6
[5,8-9]
|
α2C-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.2 – 9.4 |
pKi |
- |
1,4,7,10 |
|
⤷ |
pKi
8.2 – 9.4
[1,4,7,10]
|
α2A-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.6 – 8.9 |
pKi |
- |
1,4,7 |
|
⤷ |
pKi
7.6 – 8.9
[1,4,7]
|
α1B-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.4 – 9.0 |
pKi |
- |
5,8-9 |
|
⤷ |
pKi
7.4 – 9.0
[5,8-9]
|
α2B-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
6.8 – 8.4 |
pKi |
- |
1,4,7,10 |
|
⤷ |
pKi
6.8 – 8.4
[1,4,7,10]
|
|