AMG3054

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Ligands
AMG3054

GtoPdb Ligand ID: 9587

Compound class: Peptide or derivative

Comment: Apelin mimetic peptide agonist with reduced conformational flexibility, adopts a lactam constrained curved structure [1].

Summary
Biological activity
References
Structure
Similar ligands

References
1. Ma Y, Yue Y, Ma Y, Zhang Q, Zhou Q, Song Y, Shen Y, Li X, Ma X, Li C et al.. (2017) Structural Basis for Apelin Control of the Human Apelin Receptor. Structure, 25 (6): 858-866.e4. [PMID:28528775]

References

1. Ma Y, Yue Y, Ma Y, Zhang Q, Zhou Q, Song Y, Shen Y, Li X, Ma X, Li C et al.. (2017)
Structural Basis for Apelin Control of the Human Apelin Receptor.
Structure, 25 (6): 858-866.e4. [PMID:28528775]