|
|
|
5-HT7 receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.8 – 9.2 |
pKi |
- |
27-28 |
|
⤷ |
pKi
8.8 – 9.2
[27-28]
|
5-HT2A receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.9 |
pKi |
- |
18 |
|
⤷ |
pKi
8.9
[18]
|
5-HT7 receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.3 – 9.5 |
pKi |
- |
5,17,20 |
|
⤷ |
pKi
8.3 – 9.5
[5,17,20]
|
5-HT7 receptor
|
|
|
Mm |
Agonist |
Full agonist |
8.2 |
pKi |
- |
26 |
|
⤷ |
pKi
8.2
[26]
|
5-HT2A receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.1 |
pKi |
- |
18 |
|
⤷ |
pKi
8.1
[18]
|
5-HT1D receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.4 – 8.7 |
pKi |
- |
15,21,31 |
|
⤷ |
pKi
7.4 – 8.7
[15,21,31]
|
5-HT2B receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.0 |
pKi |
- |
30 |
|
⤷ |
pKi
8.0
[30]
|
5-HT6 receptor
|
|
|
Rn |
Agonist |
Full agonist |
6.9 – 8.4 |
pKi |
- |
8-9,24 |
|
⤷ |
pKi
6.9 – 8.4
[8-9,24]
|
5-HT1B receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.3 – 7.5 |
pKi |
- |
25,31 |
|
⤷ |
pKi
7.3 – 7.5
[25,31]
|
5-HT6 receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.4 |
pKi |
- |
19 |
|
⤷ |
pKi
7.4
[19]
|
5-HT2C receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.7 – 7.8 |
pKi |
- |
13 |
|
⤷ |
pKi
6.7 – 7.8
[13]
|
5-HT4 receptor
|
|
|
Rn |
Agonist |
Full agonist |
6.3 – 7.4 |
pKi |
- |
1,10,14 |
|
⤷ |
pKi
6.3 – 7.4
[1,10,14]
|
5-HT4 receptor
|
|
|
Mm |
Agonist |
Full agonist |
6.6 |
pKi |
- |
11 |
|
⤷ |
pKi
6.6
[11]
|
5-HT2C receptor
|
|
|
Rn |
Agonist |
Full agonist |
6.3 |
pKi |
- |
16 |
|
⤷ |
pKi
6.3
[16]
|
5-HT4 receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.6 – 6.8 |
pKi |
- |
3,6-7,22-23,29 |
|
⤷ |
pKi
5.6 – 6.8
[3,6-7,22-23,29]
|
5-HT1F receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.9 |
pKi |
- |
2 |
|
⤷ |
pKi
5.9
[2]
|
5-ht1e receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.5 – 6.2 |
pKi |
- |
2,4,12,25 |
|
⤷ |
pKi
5.5 – 6.2
[2,4,12,25]
|
|