[Ga-DOTA,Tyr3,Thr8]octreotide   Click here for help

GtoPdb Ligand ID: 5632

Synonyms: Ga-DOTA-octreotate | Ga-DOTA-TATE | Ga-DOTATATE
Compound class: Peptide or derivative
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Ligand Activity Visualisation Charts

These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.

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View interactive charts of activity data across species
References
1. Antunes P, Ginj M, Zhang H, Waser B, Baum RP, Reubi JC, Maecke H. (2007)
Are radiogallium-labelled DOTA-conjugated somatostatin analogues superior to those labelled with other radiometals?.
Eur J Nucl Med Mol Imaging, 34 (7): 982-93. [PMID:17225119]
2. Reubi JC, Schär JC, Waser B, Wenger S, Heppeler A, Schmitt JS, Mäcke HR. (2000)
Affinity profiles for human somatostatin receptor subtypes SST1-SST5 of somatostatin radiotracers selected for scintigraphic and radiotherapeutic use.
Eur J Nucl Med, 27 (3): 273-82. [PMID:10774879]