BIM 23030   Click here for help

GtoPdb Ligand ID: 2034

Comment: Cyclic peptide
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 7.7 – 7.9 pKi - 3-5
pKi 7.7 – 7.9 [3-5]
SST5 receptor Mm Agonist Full agonist 7.1 – 8.0 pKi - 1
pKi 7.1 – 8.0 [1]
SST3 receptor Hs Agonist Full agonist 7.2 – 7.8 pKi - 3,5
pKi 7.2 – 7.8 [3,5]
SST5 receptor Hs Agonist Full agonist 5.6 – 7.4 pKi - 5
pKi 5.6 – 7.4 [5]
SST2 receptor Mm Agonist Full agonist 8.2 pIC50 - 2
pIC50 8.2 [2]