galanin(D-Trp2) (pig)   Click here for help

GtoPdb Ligand ID: 6095

Compound class: Peptide
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Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
GAL2 receptor Rn Agonist Agonist 7.6 – 8.1 pKi - 2-3
pKi 7.6 – 8.1 (Ki 2.754x10-8 – 7x10-9 M) [2-3]
GAL2 receptor Hs Agonist Agonist 6.7 pKi - 1
pKi 6.7 (Ki 1.995x10-7 M) [1]
GAL1 receptor Hs Agonist Agonist 6.2 pKi - 1
pKi 6.2 (Ki 6.31x10-7 M) [1]
GAL1 receptor Rn Agonist Agonist 6.0 – 6.4 pKi - 2-3
pKi 6.0 – 6.4 (Ki 1x10-6 – 4.074x10-7 M) [2-3]
GAL3 receptor Hs Agonist Agonist <6.0 pKi - 3
pKi <6.0 (Ki >1x10-6 M) [3]
GAL3 receptor Rn Agonist Agonist <6.0 pKi - 1,3
pKi <6.0 (Ki >1x10-6 M) [1,3]
GAL2 receptor Rn Agonist Agonist 6.8 pEC50 - 2
pEC50 6.8 (EC50 1.5x10-7 M) [2]
GAL2 receptor Hs Agonist Agonist 6.5 pEC50 - 1
pEC50 6.5 (EC50 3.388x10-7 M) [1]