N-methyl-Phe-Lys-Pro-D-Cha-Cha-D-Arg-CO2H   Click here for help

GtoPdb Ligand ID: 572

Compound class: Peptide
Comment: Synthetic analogue of peptide C5a
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Ligand Activity Visualisation Charts

These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.

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View interactive charts of activity data across species
References
1. Kawai M, Quincy DA, Lane B, Mollison KW, Or YS, Luly JR, Carter GW. (1992)
Structure-function studies in a series of carboxyl-terminal octapeptide analogues of anaphylatoxin C5a.
J Med Chem, 35: 220-223. [PMID:1732540]
2. Konteatis ZD, Siciliano SJ, Van Riper G, Molineaux CJ, Pandya S, Fischer P, Rosen H, Mumford RA, Springer MS. (1994)
Development of C5a receptor antagonists. Differential loss of functional responses.
J Immunol, 153 (9): 4200-5. [PMID:7930622]