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RLF-(A11-B10)-isopeptide amideA26 (xA11-B10)   Click here for help

GtoPdb Ligand ID: 11922

Compound class: Peptide
Comment: RLF-(A11-B10)-isopeptide amideA26 (xA11-B10) is a derivative of relaxin-like factor (RLF/INSL3) in which the interchain disulphide bond is replaced with an isopeptide bond. This derivative behaves as a RXFP2 antagonist (Kd ~2 nM) [1].
Classification Click here for help
Compound class Peptide
Database Links Click here for help
Specialist databases
GPCRdb Ligand RLF-(A11-B10)-isopeptide amideA26 (xA11-B10)
Other databases
GtoPdb PubChem SID 461663477