Synonyms: Alhemo® | Anti-TFPI | concizumab-mtci | mab2021 | NN7415
concizumab is an approved drug (Health Canada (2023), FDA (2024))
Compound class:
Antibody
Comment: Concizumab is a clinical stage anti-tissue factor pathway inhibitor (TFPI) monoclonal antibody. It is a humanised IgG4 construct that was developed by Novo Nordisk as a novel therapeutic for genetic bleeding disorders [2]. Concizumab binds to the Kunitz-type protease inhibitor (KPI) 2 domain of TFPI and blocks its interaction with the active site of FXa [1]. TFPI is an endogenous anticoagulant protein whose pharmacological inhibition restores hemostasis [7].
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Classification ![]() |
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Compound class | Antibody |
Approved drug? | Yes. Health Canada (2023) | FDA (2024) | EMA (2024) |
International Nonproprietary Names ![]() |
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INN number | INN |
9636 | concizumab |
Synonyms ![]() |
Alhemo® | Anti-TFPI | concizumab-mtci | mab2021 | NN7415 |
Database Links ![]() |
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Specialist databases | |
IMGT/mAb-DB | 447 |
Other databases | |
GtoPdb PubChem SID | 434122242 |
Search PubMed clinical trials | concizumab |
Search PubMed titles | concizumab |
Search PubMed titles/abstracts | concizumab |