TCMDC-135051 [Ligand Id: 11109] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL531865
  • Plasmodium falciparum cyclin-dependent-like kinase CLK3 in Plasmodium berghei [GtoPdb: 3105]
  • Plasmodium falciparum cyclin-dependent-like kinase CLK3 in Plasmodium falciparum 3D7 [GtoPdb: 3105] [UniProtKB: Q8IIL5]
  • Plasmodium falciparum cyclin-dependent-like kinase CLK3 in Plasmodium falciparum Dd2 [GtoPdb: 3105]
  • This target only has 0 pki data point
1 CHEMBL531865_lig_chart_1 Plasmodium falciparum cyclin-dependent-like kinase CLK3 Plasmodium bergheiPlasmodium falciparum 3D7Plasmodium falciparum Dd2
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum cyclin-dependent-like kinase CLK3 in Plasmodium berghei [GtoPdb: 3105]
GtoPdb - - 6.4 pEC50 400 nM EC50 Science (2019) 365: [PMID:31467193]
Plasmodium falciparum cyclin-dependent-like kinase CLK3 in Plasmodium falciparum 3D7 [GtoPdb: 3105] [UniProtKB: Q8IIL5]
GtoPdb - - 6.49 pEC50 320 nM EC50 Science (2019) 365: [PMID:31467193]
Plasmodium falciparum cyclin-dependent-like kinase CLK3 in Plasmodium falciparum Dd2 [GtoPdb: 3105]
GtoPdb - - 6.95 pEC50 113 nM EC50 Science (2019) 365: [PMID:31467193]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]