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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BLK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 1940] [UniProtKB: P51451] | ||||||||
| GtoPdb | - | - | 6.9 | pIC50 | 125 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
| BMX non-receptor tyrosine kinase in Human [GtoPdb: 1942] [UniProtKB: P51813] | ||||||||
| GtoPdb | - | - | 7.77 | pIC50 | 17 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | - | - | 7.77 | pIC50 | 17 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
| IL2 inducible T cell kinase in Human [GtoPdb: 2046] [UniProtKB: Q08881] | ||||||||
| GtoPdb | - | - | 9.52 | pIC50 | 0.3 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 7.52 | pIC50 | 30 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
| tec protein tyrosine kinase in Human [GtoPdb: 2238] [UniProtKB: P42680] | ||||||||
| GtoPdb | - | - | 8.48 | pIC50 | 3.3 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
| TXK tyrosine kinase in Human [GtoPdb: 2268] [UniProtKB: P42681] | ||||||||
| GtoPdb | - | - | 8.85 | pIC50 | 1.4 | nM | IC50 | J Biol Chem (2015) 290: 5960-78 [PMID:25593320] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.