[des-Arg9]bradykinin [Ligand Id: 646] activity data from GtoPdb

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  • B1 receptor in Human [GtoPdb: 41] [UniProtKB: P46663]
  • B1 receptor in Mouse [GtoPdb: 41] [UniProtKB: Q61125]
Created with Highcharts 10.3.3ValuesChart context menuB1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 Mouse0246810Highcharts.com
  • B2 receptor in Human [GtoPdb: 42] [UniProtKB: P30411]
  • B2 receptor in Mouse [GtoPdb: 42] [UniProtKB: P32299]
Created with Highcharts 10.3.3ValuesChart context menuB2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 Mouse0123456Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
B1 receptor in Human [GtoPdb: 41] [UniProtKB: P46663]
GtoPdb - - 5.8 pKi - - - Eur J Pharmacol (1999) 374: 423-433 [PMID:10422787];
Br J Pharmacol (1997) 122: 393-9 [PMID:9313952]
B1 receptor in Mouse [GtoPdb: 41] [UniProtKB: Q61125]
GtoPdb - - 9.2 pKi - - - Immunopharmacology (1996) 33: 1-8 [PMID:8856107]
B2 receptor in Human [GtoPdb: 42] [UniProtKB: P30411]
GtoPdb - - 5.1 pIC50 - - - Mol Pharmacol (1994) 45: 1-8 [PMID:8302267]
B2 receptor in Mouse [GtoPdb: 42] [UniProtKB: P32299]
GtoPdb - - 5.2 pIC50 - - - Mol Pharmacol (1994) 45: 1-8 [PMID:8302267]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.