H+ [Ligand Id: 2346] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Kir1.1 in Rat [GtoPdb: 429] [UniProtKB: P35560] | ||||||||
| GtoPdb | - | - | 6.8 | pIC50 | - | - | - |
J Biol Chem (1996) 271: 17261-6 [PMID:8663367]; Am J Physiol (1995) 268: C1173-8 [PMID:7762610]; Biophys J (2003) 84: 910-21 [PMID:12547773] |
| Kir2.3 in Human [GtoPdb: 432] [UniProtKB: P48050] | ||||||||
| GtoPdb | - | - | 6.77 | pKi | - | - | - |
J Physiol (Lond.) (1999) 516 ( Pt 3): 699-710 [PMID:10200419]; J Biol Chem (2000) 275: 31573-80 [PMID:10896660] |
| GtoPdb | - | - | 7.4 | pKi | - | - | - |
Neuron (1995) 15: 1157-68 [PMID:7576658]; J Physiol (Lond.) (1999) 516 ( Pt 3): 699-710 [PMID:10200419] |
| Kir2.4 in Human [GtoPdb: 433] [UniProtKB: Q9UNX9] | ||||||||
| GtoPdb | - | - | 7.14 | pKi | - | - | - | Am J Physiol, Cell Physiol (2000) 279: C771-84 [PMID:10942728] |
| Kir4.1 in Rat [GtoPdb: 438] [UniProtKB: P49655] | ||||||||
| GtoPdb | - | - | 6.1 | pEC50 | - | - | - |
J Physiol (Lond.) (2001) 532: 359-67 [PMID:11306656]; J Biol Chem (2000) 275: 16404-7 [PMID:10764726] |
| Kir4.2 in Rat [GtoPdb: 439] [UniProtKB: Q91ZF1] | ||||||||
| GtoPdb | - | - | 7.1 | pEC50 | - | - | - | J Physiol (Lond.) (2001) 532: 359-67 [PMID:11306656] |
| TRPM5 in Human [GtoPdb: 497] [UniProtKB: Q9NZQ8] | ||||||||
| GtoPdb | - | - | 3.2 | pIC50 | 630000 | nM | IC50 | |
| TRPM7 in Human [GtoPdb: 499] [UniProtKB: Q96QT4] | ||||||||
| GtoPdb | - | - | 4.5 | pEC50 | - | - | - | J Gen Physiol (2005) 126: 137-50 [PMID:16009728] |
| TRPV1 in Human [GtoPdb: 507] [UniProtKB: Q8NER1] | ||||||||
| GtoPdb | - | - | 5.4 | pEC50 | 3980 | nM | EC50 | |
| ZAC in Human [GtoPdb: 587] [UniProtKB: Q401N2] | ||||||||
| GtoPdb | - | - | 5.6 | pEC50 | - | - | - | Biochem Pharmacol (2016) 103: 109-17 [PMID:26872532] |
| ASIC1 in Human [GtoPdb: 684] [UniProtKB: P78348] | ||||||||
| GtoPdb | - | - | 6.2 | pEC50 | ~630 | nM | EC50 | |
| GtoPdb | - | - | 6.8 | pEC50 | ~160 | nM | EC50 | |
| ASIC2 in Human [GtoPdb: 685] [UniProtKB: Q16515] | ||||||||
| GtoPdb | - | - | 5 | pEC50 | ~10000 | nM | EC50 | |
| ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3] | ||||||||
| GtoPdb | - | - | 4.3 | pEC50 | ~50000 | nM | EC50 | |
| GtoPdb | - | - | 6.7 | pEC50 | ~200 | nM | EC50 | |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
