GR 127935 [Ligand Id: 14] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL15928 (GR-127935)
  • δ receptor/Delta opioid receptor in Human [ChEMBL: CHEMBL236] [GtoPdb: 317] [UniProtKB: P41143]
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  • D1 receptor/Dopamine D1 receptor in Human [ChEMBL: CHEMBL2056] [GtoPdb: 214] [UniProtKB: P21728]
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  • D2 receptor/Dopamine D2 receptor in Human [ChEMBL: CHEMBL217] [GtoPdb: 215] [UniProtKB: P14416]
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  • D3 receptor/Dopamine D3 receptor in Human [ChEMBL: CHEMBL234] [GtoPdb: 216] [UniProtKB: P35462]
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  • D4 receptor/Dopamine D4 receptor in Human [ChEMBL: CHEMBL219] [GtoPdb: 217] [UniProtKB: P21917]
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  • D5 receptor/Dopamine D5 receptor in Human [ChEMBL: CHEMBL1850] [GtoPdb: 218] [UniProtKB: P21918]
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  • H1 receptor/Histamine H1 receptor in Human [ChEMBL: CHEMBL231] [GtoPdb: 262] [UniProtKB: P35367]
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  • κ receptor/Kappa opioid receptor in Human [ChEMBL: CHEMBL237] [GtoPdb: 318] [UniProtKB: P41145]
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  • μ receptor/Mu opioid receptor in Human [ChEMBL: CHEMBL233] [GtoPdb: 319] [UniProtKB: P35372]
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  • M1 receptor/Muscarinic acetylcholine receptor M1 in Human [ChEMBL: CHEMBL216] [GtoPdb: 13] [UniProtKB: P11229]
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  • M2 receptor/Muscarinic acetylcholine receptor M2 in Human [ChEMBL: CHEMBL211] [GtoPdb: 14] [UniProtKB: P08172]
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  • M3 receptor/Muscarinic acetylcholine receptor M3 in Human [ChEMBL: CHEMBL245] [GtoPdb: 15] [UniProtKB: P20309]
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  • M4 receptor/Muscarinic acetylcholine receptor M4 in Human [ChEMBL: CHEMBL1821] [GtoPdb: 16] [UniProtKB: P08173]
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  • M5 receptor/Muscarinic acetylcholine receptor M5 in Human [ChEMBL: CHEMBL2035] [GtoPdb: 17] [UniProtKB: P08912]
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  • 5-HT1A receptor/Serotonin 1a (5-HT1a) receptor in Human [ChEMBL: CHEMBL214] [GtoPdb: 1] [UniProtKB: P08908]
  • 5-HT1A receptor/Serotonin 1a (5-HT1a) receptor in Rat [ChEMBL: CHEMBL273] [GtoPdb: 1] [UniProtKB: P19327]
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  • 5-HT1B receptor/Serotonin 1b (5-HT1b) receptor in Human [ChEMBL: CHEMBL1898] [GtoPdb: 2] [UniProtKB: P28222]
  • 5-HT1B receptor/Serotonin 1b (5-HT1b) receptor in Rat [ChEMBL: CHEMBL3459] [GtoPdb: 2] [UniProtKB: P28564]
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  • 5-HT1D receptor/Serotonin 1d (5-HT1d) receptor in Human [ChEMBL: CHEMBL1983] [GtoPdb: 3] [UniProtKB: P28221]
  • 5-HT1D receptor/Serotonin 1d (5-HT1d) receptor in Mouse [ChEMBL: CHEMBL4297] [GtoPdb: 3] [UniProtKB: Q61224]
  • 5-HT1D receptor/Serotonin 1d (5-HT1d) receptor in Rat [ChEMBL: CHEMBL5450] [GtoPdb: 3] [UniProtKB: P28565]
  • Serotonin 1d (5-HT1d) receptor in Guinea pig [ChEMBL: CHEMBL2304407] [UniProtKB: Q60484]
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  • 5-HT2A receptor/Serotonin 2a (5-HT2a) receptor in Human [ChEMBL: CHEMBL224] [GtoPdb: 6] [UniProtKB: P28223]
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  • 5-HT2C receptor/Serotonin 2c (5-HT2c) receptor in Human [ChEMBL: CHEMBL225] [GtoPdb: 8] [UniProtKB: P28335]
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  • 5-HT4 receptor/Serotonin 4 (5-HT4) receptor in Human [ChEMBL: CHEMBL1875] [GtoPdb: 9] [UniProtKB: Q13639]
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  • 5-HT6 receptor/Serotonin 6 (5-HT6) receptor in Human [ChEMBL: CHEMBL3371] [GtoPdb: 11] [UniProtKB: P50406]
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  • 5-HT7 receptor/Serotonin 7 (5-HT7) receptor in Human [ChEMBL: CHEMBL3155] [GtoPdb: 12] [UniProtKB: P34969]
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  • SERT/Serotonin transporter in Human [ChEMBL: CHEMBL228] [GtoPdb: 928] [UniProtKB: P31645]
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  • 5-ht1e receptor in Human [GtoPdb: 4] [UniProtKB: P28566]
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  • 5-HT1F receptor in Human [GtoPdb: 5] [UniProtKB: P30939]
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  • 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor/Delta opioid receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL236] [GtoPdb: 317] [UniProtKB: P41143]
ChEMBL Affinity towards cloned Opioid receptor delta 1 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
D1 receptor/Dopamine D1 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2056] [GtoPdb: 214] [UniProtKB: P21728]
ChEMBL Binding affinity against dopamine receptor D1 B 5 pKi <10000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Affinity towards cloned Dopamine receptor D1 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
D2 receptor/Dopamine D2 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL217] [GtoPdb: 215] [UniProtKB: P14416]
ChEMBL Binding affinity against dopamine D2 receptor B 5 pKi <10000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Affinity towards cloned Dopamine receptor D2 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
D3 receptor/Dopamine D3 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL234] [GtoPdb: 216] [UniProtKB: P35462]
ChEMBL Binding affinity against dopamine D3 receptor B 5 pKi <10000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Affinity towards cloned Dopamine receptor D3 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
D4 receptor/Dopamine D4 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL219] [GtoPdb: 217] [UniProtKB: P21917]
ChEMBL Binding affinity against dopamine D4 receptor B 5 pKi <10000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Affinity towards cloned Dopamine receptor D4 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
D5 receptor/Dopamine D5 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1850] [GtoPdb: 218] [UniProtKB: P21918]
ChEMBL Affinity towards cloned Dopamine receptor D5 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
H1 receptor/Histamine H1 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL231] [GtoPdb: 262] [UniProtKB: P35367]
ChEMBL Affinity towards cloned Histamine H1 receptor B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
κ receptor/Kappa opioid receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL237] [GtoPdb: 318] [UniProtKB: P41145]
ChEMBL Affinity towards cloned Opioid receptor kappa 1 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
μ receptor/Mu opioid receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL233] [GtoPdb: 319] [UniProtKB: P35372]
ChEMBL Affinity towards cloned Opioid receptor mu 1 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
M1 receptor/Muscarinic acetylcholine receptor M1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL216] [GtoPdb: 13] [UniProtKB: P11229]
ChEMBL Affinity towards cloned Muscarinic acetylcholine receptor M1 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity against muscarinic M1 receptor B 6 pKi <1000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
M2 receptor/Muscarinic acetylcholine receptor M2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL211] [GtoPdb: 14] [UniProtKB: P08172]
ChEMBL Affinity towards cloned Muscarinic acetylcholine receptor M2 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity against muscarinic M2 receptor B 6 pKi <1000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
M3 receptor/Muscarinic acetylcholine receptor M3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL245] [GtoPdb: 15] [UniProtKB: P20309]
ChEMBL Affinity towards cloned Muscarinic acetylcholine receptor M3 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity against muscarinic M3 receptor B 6 pKi <1000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
M4 receptor/Muscarinic acetylcholine receptor M4 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1821] [GtoPdb: 16] [UniProtKB: P08173]
ChEMBL Affinity towards cloned Muscarinic acetylcholine receptor M4 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
M5 receptor/Muscarinic acetylcholine receptor M5 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2035] [GtoPdb: 17] [UniProtKB: P08912]
ChEMBL Affinity towards cloned Muscarinic acetylcholine receptor M5 B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
5-HT1A receptor/Serotonin 1a (5-HT1a) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL214] [GtoPdb: 1] [UniProtKB: P08908]
ChEMBL In vitro binding affinity towards cloned human 5-HT1A receptor using [3H]5-carboximidotryptamine as radioligand B 7.1 pKi 80 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Affinity for 5-hydroxytryptamine 1A receptor subtype B 7.14 pKi 72 nM Ki Bioorg Med Chem Lett (1997) 7: 3183-3188
ChEMBL Affinity towards cloned human 5-hydroxytryptamine 1A receptor B 7.15 pKi 70 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
GtoPdb - - 7.2 pKi - - - J Med Chem (1997) 40: 3974-8 [PMID:9397179];
Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567]
5-HT1A receptor/Serotonin 1a (5-HT1a) receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL273] [GtoPdb: 1] [UniProtKB: P19327]
ChEMBL Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus with [3H]8-OH-DPAT B 6.5 pKi 316.23 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Inhibition activity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using radio binding assays B 6.37 pIC50 425 nM IC50 J Med Chem (2000) 43: 517-525 [PMID:10669578]
ChEMBL Binding affinity towards 5-hydroxytryptamine 1A receptor in rat frontal cortex using [125I]iodocyanopindolol as radio-ligand. B 6.44 pIC50 360 nM IC50 J Med Chem (2000) 43: 1149-1157 [PMID:10737747]
5-HT1B receptor/Serotonin 1b (5-HT1b) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1898] [GtoPdb: 2] [UniProtKB: P28222]
ChEMBL In vitro binding affinity towards cloned human 5-HT1B receptor using [3H]5-carboximidotryptamine as radioligand B 8.37 pKi 4.31 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity for human 5-hydroxytryptamine 1B receptor B 9 pKi 1 nM Ki J Med Chem (1998) 41: 1218-1235 [PMID:9548813]
GtoPdb - - 9.2 pKi - - - Eur J Pharmacol (1999) 380: 171-81 [PMID:10513577]
GtoPdb - - 9.8 pKi - - - J Med Chem (1997) 40: 3974-8 [PMID:9397179];
Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567];
Br J Pharmacol (1998) 125: 202-8 [PMID:9776361];
Eur J Pharmacol (1996) 314: 365-72 [PMID:8957260];
J Med Chem (1998) 41: 1218-35 [PMID:9548813]
ChEMBL Affinity for 5-hydroxytryptamine 1B receptor subtype B 9.85 pKi 0.14 nM Ki Bioorg Med Chem Lett (1997) 7: 3183-3188
ChEMBL Affinity towards cloned human 5-hydroxytryptamine 1B receptor B 9.85 pKi 0.14 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
5-HT1B receptor/Serotonin 1b (5-HT1b) receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3459] [GtoPdb: 2] [UniProtKB: P28564]
ChEMBL In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindolol B 8.5 pKi 3.16 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Inhibition affinity against 5-HT-1B receptor in rat frontal cortex using radio binding assay B 8.8 pIC50 1.6 nM IC50 J Med Chem (2000) 43: 517-525 [PMID:10669578]
ChEMBL Binding affinity towards 5-hydroxytryptamine 1B receptor in rat frontal cortex using [125I]iodocyanopindolol as radio-ligand. B 8.8 pIC50 1.6 nM IC50 J Med Chem (2000) 43: 1149-1157 [PMID:10737747]
5-HT1D receptor/Serotonin 1d (5-HT1d) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1983] [GtoPdb: 3] [UniProtKB: P28221]
ChEMBL In vitro binding affinity towards cloned human 5-HT1D receptor using [3H]5-carboximidotryptamine as radioligand B 7.91 pKi 12.3 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity for human 5-hydroxytryptamine 1D receptor B 8.6 pKi 2.51 nM Ki J Med Chem (1998) 41: 1218-1235 [PMID:9548813]
GtoPdb - - 8.6 pKi - - - Mol Pharmacol (1996) 50: 1567-80 [PMID:8967979]
ChEMBL Binding affinity against 5-hydroxytryptamine 1D receptor alpha B 8.9 pKi 1.26 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
GtoPdb - - 9.1 pKi - - - J Med Chem (1997) 40: 3974-8 [PMID:9397179];
Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567];
Br J Pharmacol (1998) 125: 202-8 [PMID:9776361];
Eur J Pharmacol (1996) 314: 365-72 [PMID:8957260];
J Med Chem (1998) 41: 1218-35 [PMID:9548813]
ChEMBL Affinity for 5-hydroxytryptamine 1D receptor subtype B 9.15 pKi 0.7 nM Ki Bioorg Med Chem Lett (1997) 7: 3183-3188
ChEMBL Affinity towards cloned human 5-hydroxytryptamine 1D receptor B 9.15 pKi 0.7 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity against 5-hydroxytryptamine 1D receptor beta B 9.9 pKi 0.13 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
ChEMBL Inhibition affinity against 5-HT-1D receptor in bovine caudate nucleus using radio binding assay B 7.28 pIC50 52 nM IC50 J Med Chem (2000) 43: 517-525 [PMID:10669578]
5-HT1D receptor/Serotonin 1d (5-HT1d) receptor in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4297] [GtoPdb: 3] [UniProtKB: Q61224]
ChEMBL Tested for 5-hydroxytryptamine receptor uptake F 5 pKi <10000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
5-HT1D receptor/Serotonin 1d (5-HT1d) receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5450] [GtoPdb: 3] [UniProtKB: P28565]
ChEMBL Binding affinity towards 5-hydroxytryptamine 1D receptor in rat frontal cortex using [125I]iodocyanopindolol as radio-ligand. B 7.28 pIC50 53 nM IC50 J Med Chem (2000) 43: 1149-1157 [PMID:10737747]
Serotonin 1d (5-HT1d) receptor in Guinea pig (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2304407] [UniProtKB: Q60484]
ChEMBL In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergine B 8.5 pKi 3.16 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
5-HT2A receptor/Serotonin 2a (5-HT2a) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL224] [GtoPdb: 6] [UniProtKB: P28223]
ChEMBL In vitro binding affinity towards cloned human 5-HT2A receptor using [3H]5-carboximidotryptamine as radioligand B 7.37 pKi 42.7 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
ChEMBL Binding affinity for human 5-hydroxytryptamine 2A receptor B 7.8 pKi 15.85 nM Ki J Med Chem (1998) 41: 1218-1235 [PMID:9548813]
GtoPdb - - 7.8 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567];
J Med Chem (1998) 41: 1218-35 [PMID:9548813]
5-HT2C receptor/Serotonin 2c (5-HT2c) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL225] [GtoPdb: 8] [UniProtKB: P28335]
ChEMBL In vitro binding affinity towards cloned human 5-HT2C receptor using [3H]5-carboximidotryptamine as radioligand B 6.98 pKi 105 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
GtoPdb - - 7 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567]
5-HT3E/5-HT3B/5-HT3A/5-HT3D/5-HT3C/Serotonin 3 (5-HT3) receptor in Human (target type: PROTEIN COMPLEX GROUP) [ChEMBL: CHEMBL2094132] [GtoPdb: 377, 374, 373, 376, 375] [UniProtKB: A5X5Y0, O95264, P46098, Q70Z44, Q8WXA8]
ChEMBL Binding affinity against the 5-hydroxytryptamine 3 receptor B 5.2 pKi 6309.57 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
5-HT4 receptor/Serotonin 4 (5-HT4) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1875] [GtoPdb: 9] [UniProtKB: Q13639]
ChEMBL Binding affinity against 5-hydroxytryptamine 4 receptor B 5 pKi <10000 nM Ki J Med Chem (1994) 37: 2253-2257 [PMID:8057272]
5-HT6 receptor/Serotonin 6 (5-HT6) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3371] [GtoPdb: 11] [UniProtKB: P50406]
ChEMBL In vitro binding affinity towards cloned human 5-HT6 receptor using [3H]5-carboximidotryptamine as radioligand B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
GtoPdb - - 5.8 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567]
5-HT7 receptor/Serotonin 7 (5-HT7) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3155] [GtoPdb: 12] [UniProtKB: P34969]
ChEMBL In vitro binding affinity towards cloned human 5-HT7 receptor using [3H]5-carboximidotryptamine as radioligand B 5 pKi >10000 nM Ki Bioorg Med Chem Lett (2005) 15: 4786-4789 [PMID:16143528]
SERT/Serotonin transporter in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL228] [GtoPdb: 928] [UniProtKB: P31645]
ChEMBL Inhibition of 5-hydroxytryptamine reuptake B 6 pIC50 1000 nM IC50 J Med Chem (2000) 43: 517-525 [PMID:10669578]
5-ht1e receptor in Human [GtoPdb: 4] [UniProtKB: P28566]
GtoPdb - - 5.4 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567]
5-HT1F receptor in Human [GtoPdb: 5] [UniProtKB: P30939]
GtoPdb - - 7.2 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567];
Naunyn Schmiedebergs Arch Pharmacol (2005) 371: 169-77 [PMID:15900510]
5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
GtoPdb - - 6.2 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1997) 356: 312-20 [PMID:9303567]

ChEMBL data shown on this page come from version 34:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]