compound 6 [PMID: 34333981] [Ligand Id: 11893] activity data from GtoPdb

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  • AP2 associated kinase 1 in Human [GtoPdb: 1921] [UniProtKB: Q2M2I8]
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  • BMP2 inducible kinase in Human [GtoPdb: 1941] [UniProtKB: Q9NSY1]
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  • serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716]
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  • TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2]
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  • tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
AP2 associated kinase 1 in Human [GtoPdb: 1921] [UniProtKB: Q2M2I8]
GtoPdb - - 7.1 pIC50 80 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
BMP2 inducible kinase in Human [GtoPdb: 1941] [UniProtKB: Q9NSY1]
GtoPdb - - 7.42 pIC50 38 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716]
GtoPdb - - 7.06 pIC50 88 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2]
GtoPdb - - 7.18 pIC50 66 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597]
GtoPdb - - 7.17 pIC50 67 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.