GSK2833503A [Ligand Id: 10284] activity data from GtoPdb

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  • TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
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  • TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
GtoPdb Measuring whole-cell current by patch-clamp in HEK cells expressing hTRPC3 with cation flux activated by OAG. - 7.68 pIC50 21 nM IC50 Proc Natl Acad Sci USA (2014) 111: 1551-6 [PMID:24453217]
TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210]
GtoPdb Measuring whole-cell current by patch-clamp in HEK cells expressing hTRPC6 with cation flux activated by OAG. - 8.52 pIC50 3 nM IC50 Proc Natl Acad Sci USA (2014) 111: 1551-6 [PMID:24453217]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.