JAK3 inhibitor 32 [Ligand Id: 10156] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | - | - | 5.57 | pIC50 | 2703 | nM | IC50 | J Med Chem (2018) 61: 10665-10699 [PMID:30423248] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 5.52 | pIC50 | 3012 | nM | IC50 | J Med Chem (2018) 61: 10665-10699 [PMID:30423248] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 7.96 | pIC50 | 11 | nM | IC50 | J Med Chem (2018) 61: 10665-10699 [PMID:30423248] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | - | - | 5 | pIC50 | >10000 | nM | IC50 | J Med Chem (2018) 61: 10665-10699 [PMID:30423248] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
