KBP-7018 [Ligand Id: 9691] activity data from GtoPdb

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  • platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619]
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  • KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721]
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  • ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619]
GtoPdb - - 7.6 pIC50 25 nM IC50 ACS Med Chem Lett (2017) 8: 1142-1147 [PMID:29152045]
KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721]
GtoPdb - - 8 pIC50 10 nM IC50 ACS Med Chem Lett (2017) 8: 1142-1147 [PMID:29152045]
ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949]
GtoPdb - - 8.12 pIC50 7.6 nM IC50 ACS Med Chem Lett (2017) 8: 1142-1147 [PMID:29152045]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.