ML324 [Ligand Id: 9584] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1398529
  • lysine demethylase 4A in Human [GtoPdb: 2675] [UniProtKB: O75164]
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  • lysine demethylase 4E in Human [GtoPdb: 2679] [UniProtKB: B2RXH2]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
lysine demethylase 4A in Human [GtoPdb: 2675] [UniProtKB: O75164]
GtoPdb - - 6 pIC50 <1000 nM IC50 Probe Reports from the NIH Molecular Libraries Program (2010) : [PMID:24260783]
lysine demethylase 4E in Human [GtoPdb: 2679] [UniProtKB: B2RXH2]
GtoPdb - - 6.04 pIC50 920 nM IC50 Probe Reports from the NIH Molecular Libraries Program (2010) : [PMID:24260783]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]