compound II [PMID: 21329883] [Ligand Id: 9579] activity data from GtoPdb

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  • inhibitor of nuclear factor kappa B kinase subunit epsilon in Human [GtoPdb: 2040] [UniProtKB: Q14164]
Created with Highcharts 10.3.3ValuesChart context menuinhibitor of nuclear factor kappa B kinase subunit epsilonpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2]
Created with Highcharts 10.3.3ValuesChart context menuTANK binding kinase 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
inhibitor of nuclear factor kappa B kinase subunit epsilon in Human [GtoPdb: 2040] [UniProtKB: Q14164]
GtoPdb In a biochemical assay using purified recombinant enzyme. - 7.23 pIC50 59 nM IC50 Mol Cell (2011) 41: 458-70 [PMID:21329883]
TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2]
GtoPdb In a biochemical assay using purified recombinant enzyme. - 7.89 pIC50 13 nM IC50 Mol Cell (2011) 41: 458-70 [PMID:21329883]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.