BLU-9931 [Ligand Id: 8862] activity data from GtoPdb

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  • fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362]
Created with Highcharts 10.3.3ValuesChart context menufibroblast growth factor receptor 1pKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
  • fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802]
Created with Highcharts 10.3.3ValuesChart context menufibroblast growth factor receptor 2pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607]
Created with Highcharts 10.3.3ValuesChart context menufibroblast growth factor receptor 3pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455]
Created with Highcharts 10.3.3ValuesChart context menufibroblast growth factor receptor 4pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362]
GtoPdb - - 6.23 pIC50 591 nM IC50 Cancer Discov (2015) 5: 424-37 [PMID:25776529]
fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802]
GtoPdb - - 6.31 pIC50 493 nM IC50 Cancer Discov (2015) 5: 424-37 [PMID:25776529]
fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607]
GtoPdb - - 6.82 pIC50 150 nM IC50 Cancer Discov (2015) 5: 424-37 [PMID:25776529]
fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455]
GtoPdb - - 8.52 pIC50 3 nM IC50 Cancer Discov (2015) 5: 424-37 [PMID:25776529]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.