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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
ribosomal protein S6 kinase A6 in Human [GtoPdb: 1530] [UniProtKB: Q9UK32] | ||||||||
GtoPdb | - | - | 8 | pIC50 | 10 | nM | IC50 | J Med Chem (2009) 52: 379-88 [PMID:19143567] |
aurora kinase A in Human [GtoPdb: 1936] [UniProtKB: O14965] | ||||||||
GtoPdb | - | - | 8.52 | pIC50 | ~3 | nM | IC50 | J Med Chem (2009) 52: 379-88 [PMID:19143567] |
aurora kinase B in Human [GtoPdb: 1937] [UniProtKB: Q96GD4] | ||||||||
GtoPdb | - | - | 8.52 | pIC50 | ~3 | nM | IC50 | J Med Chem (2009) 52: 379-88 [PMID:19143567] |
Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
GtoPdb | - | - | 8.92 | pIC50 | 1.2 | nM | IC50 | J Med Chem (2009) 52: 379-88 [PMID:19143567] |
Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
GtoPdb | - | - | 8.96 | pIC50 | 1.1 | nM | IC50 | J Med Chem (2009) 52: 379-88 [PMID:19143567] |
serine/threonine kinase 17a in Human [GtoPdb: 2214] [UniProtKB: Q9UEE5] | ||||||||
GtoPdb | - | - | 8 | pIC50 | 10 | nM | IC50 | J Med Chem (2009) 52: 379-88 [PMID:19143567] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.