vMIP-II [Ligand Id: 768] activity data from GtoPdb

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  • CCR1 in Human [GtoPdb: 58] [UniProtKB: P32246]
Created with Highcharts 10.3.3ValuesChart context menuCCR1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
Created with Highcharts 10.3.3ValuesChart context menuCCR2pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • CCR5 in Human [GtoPdb: 62] [UniProtKB: P51681]
Created with Highcharts 10.3.3ValuesChart context menuCCR5pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • CCR8 in Human [GtoPdb: 65] [UniProtKB: P51685]
Created with Highcharts 10.3.3ValuesChart context menuCCR8pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • CXCR4 in Human [GtoPdb: 71] [UniProtKB: P61073]
Created with Highcharts 10.3.3ValuesChart context menuCXCR4pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CCR1 in Human [GtoPdb: 58] [UniProtKB: P32246]
GtoPdb - - 8.1 pIC50 - - - Science (1997) 277: 1656-9 [PMID:9287217]
CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
GtoPdb - - 9.1 pIC50 - - - Science (1997) 277: 1656-9 [PMID:9287217]
CCR5 in Human [GtoPdb: 62] [UniProtKB: P51681]
GtoPdb - - 8.3 pIC50 - - - Science (1997) 277: 1656-9 [PMID:9287217]
CCR8 in Human [GtoPdb: 65] [UniProtKB: P51685]
GtoPdb - - 8.1 pIC50 - - - J Biol Chem (1999) 274: 21569-74 [PMID:10419462]
CXCR4 in Human [GtoPdb: 71] [UniProtKB: P61073]
GtoPdb - - 8.2 pIC50 - - - Science (1997) 277: 1656-9 [PMID:9287217]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.