compound 36 [PMID: 24000170] [Ligand Id: 7521] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • bromodomain containing 2 in Human [GtoPdb: 1944] [UniProtKB: P25440]
There should be some charts here, you may need to enable JavaScript!
  • bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
There should be some charts here, you may need to enable JavaScript!
  • bromodomain containing 3 in Human [GtoPdb: 2725] [UniProtKB: Q15059]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 2 in Human [GtoPdb: 1944] [UniProtKB: P25440]
GtoPdb - - 6 pIC50 1000 nM IC50 ChemMedChem (2014) 9: 580-9 [PMID:24000170]
bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
GtoPdb - - 6.2 pIC50 631 nM IC50 ChemMedChem (2014) 9: 580-9 [PMID:24000170]
bromodomain containing 3 in Human [GtoPdb: 2725] [UniProtKB: Q15059]
GtoPdb - - 6.3 pIC50 501 nM IC50 ChemMedChem (2014) 9: 580-9 [PMID:24000170]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.