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ChEMBL ligand: CHEMBL1740 (Vaponefrin, Racepinefrine, Racepinephrine) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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α2B-adrenoceptor in Human [GtoPdb: 26] [UniProtKB: P18089] | ||||||||
GtoPdb | - | - | 6.2 | pKi | - | - | - | Biochem Pharmacol (1998) 55: 1035-43 [PMID:9605427] |
α2C-adrenoceptor in Human [GtoPdb: 27] [UniProtKB: P18825] | ||||||||
GtoPdb | - | - | 6.2 | pKi | - | - | - | Biochem Pharmacol (1998) 55: 1035-43 [PMID:9605427] |
β1-adrenoceptor in Human [GtoPdb: 28] [UniProtKB: P08588] | ||||||||
GtoPdb | - | - | 6 | pKi | - | - | - | Proc Natl Acad Sci USA (1988) 85: 9494-8 [PMID:2849109] |
β3-adrenoceptor in Human [GtoPdb: 30] [UniProtKB: P13945] | ||||||||
GtoPdb | - | - | 4.7 | pKi | - | - | - |
Eur J Pharmacol (1995) 291: 359-66 [PMID:8719421]; Mol Pharmacol (1993) 44: 1094-104 [PMID:7903415]; Naunyn Schmiedebergs Arch Pharmacol (2004) 369: 151-9 [PMID:14730417] |
β3-adrenoceptor in Mouse [GtoPdb: 30] [UniProtKB: P25962] | ||||||||
GtoPdb | - | - | 5.3 | pKi | - | - | - | Eur J Pharmacol (1995) 291: 359-66 [PMID:8719421] |
β3-adrenoceptor in Rat [GtoPdb: 30] [UniProtKB: P26255] | ||||||||
GtoPdb | - | - | 5.3 | pKi | - | - | - | Eur J Pharmacol (1995) 291: 359-66 [PMID:8719421] |
ChEMBL data shown on this page come from version 28:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]