eratrectinib [Ligand Id: 14070] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| neurotrophic receptor tyrosine kinase 1 in Human [GtoPdb: 1817] [UniProtKB: P04629] | ||||||||
| GtoPdb | - | - | 8.37 | pIC50 | 4.23 | nM | IC50 | WO2019233461A1. Tropomyosin receptor kinase inhibitor, preparation method therefor and use thereof (2019) |
| neurotrophic receptor tyrosine kinase 2 in Human [GtoPdb: 1818] [UniProtKB: Q16620] | ||||||||
| GtoPdb | - | - | 9.24 | pIC50 | 0.57 | nM | IC50 | WO2019233461A1. Tropomyosin receptor kinase inhibitor, preparation method therefor and use thereof (2019) |
| neurotrophic receptor tyrosine kinase 3 in Human [GtoPdb: 1819] [UniProtKB: Q16288] | ||||||||
| GtoPdb | - | - | 9.6 | pIC50 | 0.25 | nM | IC50 | WO2019233461A1. Tropomyosin receptor kinase inhibitor, preparation method therefor and use thereof (2019) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
