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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CYP1A2 in Human [GtoPdb: 1319] [UniProtKB: P05177] | ||||||||
| GtoPdb | - | - | 5.5 | pKi | 3180 | nM | Ki | Pharmacol Res Perspect (2024) 12: e70002 [PMID:39210686] |
| CYP2D6 in Human [GtoPdb: 1329] [UniProtKB: P10635] | ||||||||
| GtoPdb | - | - | 5.17 | pKi | 6770 | nM | Ki | Pharmacol Res Perspect (2024) 12: e70002 [PMID:39210686] |
| CYP3A4 in Human [GtoPdb: 1337] [UniProtKB: P08684] | ||||||||
| GtoPdb | - | - | 5.62 | pKi | 2380 | nM | Ki | Pharmacol Res Perspect (2024) 12: e70002 [PMID:39210686] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.