elenestinib [Ligand Id: 12357] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor alpha in Human [GtoPdb: 1803] [UniProtKB: P16234] | ||||||||
| GtoPdb | Biochemical inhibition assay, using PDGFRαD842V | - | 8.35 | pIC50 | <4.5 | nM | IC50 | WO2020210293A1. Pyrrolotriazine derivatives for treating kit- and pdgfra-mediated diseases (2020) |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | Biochemical inhibition assay, using KITD816V | - | 8.35 | pIC50 | <4.5 | nM | IC50 | WO2020210293A1. Pyrrolotriazine derivatives for treating kit- and pdgfra-mediated diseases (2020) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
