XY-06-007 [Ligand Id: 12141] activity data from GtoPdb

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  • bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
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  • polo like kinase 1 in Human [GtoPdb: 2168] [UniProtKB: P53350]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
GtoPdb - - 6.6 pIC50 254 nM IC50 Eur J Med Chem (2022) 227: 113922 [PMID:34700270]
polo like kinase 1 in Human [GtoPdb: 2168] [UniProtKB: P53350]
GtoPdb - - 6.01 pIC50 985 nM IC50 Eur J Med Chem (2022) 227: 113922 [PMID:34700270]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.