BAY-545 [Ligand Id: 11224] activity data from GtoPdb

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  • A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275]
  • A2B receptor in Mouse [GtoPdb: 20] [UniProtKB: Q60614]
  • A2B receptor in Rat [GtoPdb: 20] [UniProtKB: P29276]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275]
GtoPdb - - 7.01 pKi 97 nM Ki Eur J Med Chem (2019) 163: 763-778 [PMID:30576906]
A2B receptor in Mouse [GtoPdb: 20] [UniProtKB: Q60614]
GtoPdb - - 6.4 pIC50 400 nM IC50 Eur J Med Chem (2019) 163: 763-778 [PMID:30576906]
A2B receptor in Rat [GtoPdb: 20] [UniProtKB: P29276]
GtoPdb - - 6.55 pIC50 280 nM IC50 Eur J Med Chem (2019) 163: 763-778 [PMID:30576906]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.