vimseltinib [Ligand Id: 11190] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor alpha in Human [GtoPdb: 1803] [UniProtKB: P16234] | ||||||||
| GtoPdb | - | - | 6 | pIC50 | >1000 | nM | IC50 | WO2014145025A2. 2-aminopyrimidin-6-ones and analogs exhibiting anti-cancer and anti-proliferative activities (2014) |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | - | - | 7 | pIC50 | 100 | nM | IC50 | WO2014145025A2. 2-aminopyrimidin-6-ones and analogs exhibiting anti-cancer and anti-proliferative activities (2014) |
| colony stimulating factor 1 receptor in Human [GtoPdb: 1806] [UniProtKB: P07333] | ||||||||
| GtoPdb | - | - | 8 | pIC50 | <10 | nM | IC50 | WO2014145025A2. 2-aminopyrimidin-6-ones and analogs exhibiting anti-cancer and anti-proliferative activities (2014) |
| GtoPdb | - | - | 8.43 | pIC50 | 3.7 | nM | IC50 | Bioorg Med Chem Lett (2022) 74: 128928 [PMID:35961460] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
