ibcasertib [Ligand Id: 10475] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor alpha in Human [GtoPdb: 1803] [UniProtKB: P16234] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 9 | pIC50 | 1 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 7.03 | pIC50 | 93 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 8.4 | pIC50 | 4 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| colony stimulating factor 1 receptor in Human [GtoPdb: 1806] [UniProtKB: P07333] | ||||||||
| GtoPdb | - | - | 8.15 | pIC50 | 7 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| fms related receptor tyrosine kinase 1 in Human [GtoPdb: 1812] [UniProtKB: P17948] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 8.1 | pIC50 | 8 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 8.15 | pIC50 | 7 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| fms related receptor tyrosine kinase 4 in Human [GtoPdb: 1814] [UniProtKB: P35916] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 8.05 | pIC50 | 9 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
| aurora kinase B in Human [GtoPdb: 1937] [UniProtKB: Q96GD4] | ||||||||
| GtoPdb | Inhibition in a biochemical assay. | - | 8.05 | pIC50 | 9 | nM | IC50 | Cancer Sci (2017) 108: 469-477 [PMID:28004478] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
