tonantzitlolone [Ligand Id: 10287] activity data from GtoPdb

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  • TRPC4 in Human [GtoPdb: 489] [UniProtKB: Q9UBN4]
Created with Highcharts 10.3.3ValuesChart context menuTRPC4pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • TRPC5 in Human [GtoPdb: 490] [UniProtKB: Q9UL62]
Created with Highcharts 10.3.3ValuesChart context menuTRPC5pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPC4 in Human [GtoPdb: 489] [UniProtKB: Q9UBN4]
GtoPdb - - 6.91 pEC50 123 nM EC50 Br J Pharmacol (2018) 175: 3361-3368 [PMID:29859013]
TRPC5 in Human [GtoPdb: 490] [UniProtKB: Q9UL62]
GtoPdb - - 7.08 pEC50 83 nM EC50 Br J Pharmacol (2018) 175: 3361-3368 [PMID:29859013]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.