AM10257 [Ligand Id: 10177] activity data from GtoPdb

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  • CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
Created with Highcharts 10.3.3ValuesChart context menuCB2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
GtoPdb Antagonism of [3H]CP55940 binding to human CB2. - 10.12 pKi 0.08 nM Ki Cell (2019) 176: 459-467.e13 [PMID:30639103]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.