kinase inhibitor 2 [PMID: 30199702] [Ligand Id: 10081] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493] | ||||||||
| GtoPdb | CDK1/cyclin B | - | 7.15 | pIC50 | 70 | nM | IC50 | Eur J Med Chem (2018) 158: 1-6 [PMID:30199702] |
| cyclin dependent kinase 2 in Human [GtoPdb: 1973] [UniProtKB: P24941] | ||||||||
| GtoPdb | CDK2/cyclin A | - | 7.17 | pIC50 | 68 | nM | IC50 | Eur J Med Chem (2018) 158: 1-6 [PMID:30199702] |
| cyclin dependent kinase 5 in Human [GtoPdb: 1977] [UniProtKB: Q00535] | ||||||||
| GtoPdb | CDK5/p25 | - | 7.3 | pIC50 | 50 | nM | IC50 | Eur J Med Chem (2018) 158: 1-6 [PMID:30199702] |
| cyclin dependent kinase 9 in Human [GtoPdb: 1981] [UniProtKB: P50750] | ||||||||
| GtoPdb | CDK9/cyclin T | - | 7.31 | pIC50 | 49 | nM | IC50 | Eur J Med Chem (2018) 158: 1-6 [PMID:30199702] |
| CDC like kinase 4 in Human [GtoPdb: 1993] [UniProtKB: Q9HAZ1] | ||||||||
| GtoPdb | - | - | 7.05 | pIC50 | 89 | nM | IC50 | Eur J Med Chem (2018) 158: 1-6 [PMID:30199702] |
| dual specificity tyrosine phosphorylation regulated kinase 3 in Human [GtoPdb: 2012] [UniProtKB: O43781] | ||||||||
| GtoPdb | - | - | 6.42 | pIC50 | 380 | nM | IC50 | Eur J Med Chem (2018) 158: 1-6 [PMID:30199702] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
