isoquinoline 17 [PMID: 30122040] [Ligand Id: 10071] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| kelch like ECH-associated protein 1 in Human [GtoPdb: 2757] [UniProtKB: Q14145] | ||||||||
| GtoPdb | Binding to hKEAP1 by SPR. | - | 6.99 | pKd | 102 | nM | Kd | J Med Chem (2018) 61: 8029-8047 [PMID:30122040] |
| GtoPdb | Measured by fluorescence anisotropy. | - | 7.22 | pIC50 | 60 | nM | IC50 | J Med Chem (2018) 61: 8029-8047 [PMID:30122040] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
