azelaprag [Ligand Id: 10061] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| apelin receptor in Human [GtoPdb: 36] [UniProtKB: P35414] | ||||||||
| GtoPdb | Measuring ligand-induced [35S]GTPyS Binding in membranes prepared fron CHO cells stably expressing human apelin receptor. | - | 9.49 | pEC50 | 0.32 | nM | EC50 |
WO2016187308A1. Triazole agonists of the apj receptor (2016); JCI Insight (2020) 5: [PMID:32208384] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
