PF-04634817 [Ligand Id: 9979] activity data from GtoPdb

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  • CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
Created with Highcharts 10.3.3ValuesChart context menuCCR2pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
GtoPdb Whole cell binding assay measuring displacement of [125I]MCP-1 from CCR2 by PF-04634817 in human peripheral blood mononuclear cells. - 8.43 pIC50 3.68 nM IC50 US8293903B2. 3-aminocyclopentanecarboxamides as chemokine receptor agonists. (2012)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.