voruciclib [Ligand Id: 9923] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493] | ||||||||
| GtoPdb | Inhibition of CDK1/cyclinB | - | 7.6 | pIC50 | 25 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| cyclin dependent kinase 2 in Human [GtoPdb: 1973] [UniProtKB: P24941] | ||||||||
| GtoPdb | Inhibition of CDK2/cyclinA | - | 6.74 | pIC50 | 180 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802] | ||||||||
| GtoPdb | Inhibition of CDK4/cyclinD1. | - | 7.05 | pIC50 | 90 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| cyclin dependent kinase 5 in Human [GtoPdb: 1977] [UniProtKB: Q00535] | ||||||||
| GtoPdb | Inhibition of CDK5/cyclin p35 (CDK5R1). | - | 6.68 | pIC50 | 210 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534] | ||||||||
| GtoPdb | Inhibition of CDK6/cyclinD3. | - | 6.68 | pIC50 | 210 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| cyclin dependent kinase 8 in Human [GtoPdb: 1980] [UniProtKB: P49336] | ||||||||
| GtoPdb | Inhibition of CDK8/cyclinC. | - | 7.92 | pIC50 | 12 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| cyclin dependent kinase 9 in Human [GtoPdb: 1981] [UniProtKB: P50750] | ||||||||
| GtoPdb | Inhibition of CDK9/cyclinT. | - | 7.66 | pIC50 | 22 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| casein kinase 1 gamma 1 in Human [GtoPdb: 1999] [UniProtKB: Q9HCP0] | ||||||||
| GtoPdb | - | - | 6.96 | pIC50 | 110 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| dual specificity tyrosine phosphorylation regulated kinase 1B in Human [GtoPdb: 2010] [UniProtKB: Q9Y463] | ||||||||
| GtoPdb | - | - | 7.03 | pIC50 | 94 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| glycogen synthase kinase 3 alpha in Human [GtoPdb: 2029] [UniProtKB: P49840] | ||||||||
| GtoPdb | - | - | 7.77 | pIC50 | 17 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| glycogen synthase kinase 3 beta in Human [GtoPdb: 2030] [UniProtKB: P49841] | ||||||||
| GtoPdb | - | - | 7.15 | pIC50 | 71 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| LIM domain kinase 1 in Human [GtoPdb: 2054] [UniProtKB: P53667] | ||||||||
| GtoPdb | - | - | 7.66 | pIC50 | 22 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| mitogen-activated protein kinase kinase 2 in Human [GtoPdb: 2063] [UniProtKB: P36507] | ||||||||
| GtoPdb | - | - | 7.06 | pIC50 | 87 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
| Pim-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2158] [UniProtKB: P11309] | ||||||||
| GtoPdb | - | - | 7.14 | pIC50 | 72 | nM | IC50 | PLoS ONE (2015) 10: e0143685 [PMID:26606677] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
