tucatinib [Ligand Id: 9922] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | Inhibition of enzyme activity in a biochemical assay. | - | 6.35 | pIC50 | 449 | nM | IC50 | Mol Cancer Ther (2020) 19: 976-987 [PMID:32241871] |
| erb-b2 receptor tyrosine kinase 4 in Human [GtoPdb: 1799] [UniProtKB: Q15303] | ||||||||
| GtoPdb | Inhibition of enzyme activity in a biochemical assay. | - | 6.51 | pIC50 | 310 | nM | IC50 | Mol Cancer Ther (2020) 19: 976-987 [PMID:32241871] |
| erb-b2 receptor tyrosine kinase 2 in Human [GtoPdb: 2019] [UniProtKB: P04626] | ||||||||
| GtoPdb | Inhibition of enzyme activity in a biochemical assay. | - | 8.16 | pIC50 | 6.9 | nM | IC50 | Mol Cancer Ther (2020) 19: 976-987 [PMID:32241871] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
