H05 [Ligand Id: 9880] activity data from GtoPdb

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  • 5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
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  • NET in Rat [GtoPdb: 926]
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  • SERT in Rat [GtoPdb: 928] [UniProtKB: P31652]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
GtoPdb - - 7.22 pIC50 60.37 nM IC50 J Pharmacol Exp Ther (2018) 365: 624-635 [PMID:29615471]
NET in Rat [GtoPdb: 926]
GtoPdb - - 8.17 pKi 6.72 nM Ki J Pharmacol Exp Ther (2018) 365: 624-635 [PMID:29615471]
SERT in Rat [GtoPdb: 928] [UniProtKB: P31652]
GtoPdb - - 8.32 pKi 4.81 nM Ki J Pharmacol Exp Ther (2018) 365: 624-635 [PMID:29615471]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.