GS-458967 [Ligand Id: 9858] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Nav1.5 in Human [GtoPdb: 582] [UniProtKB: Q14524] | ||||||||
| GtoPdb | - | - | 6.89 | pIC50 | 130 | nM | IC50 |
Bioorg Med Chem Lett (2016) 26: 3202-3206 [PMID:27080178]; Br J Pharmacol (2018) 175: 2470-2482 [PMID:29582428] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
