compound 47 [PMID: 28737909] [Ligand Id: 9646] activity data from GtoPdb

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  • component of inhibitor of nuclear factor kappa B kinase complex in Human [GtoPdb: 1989] [UniProtKB: O15111]
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  • inhibitor of nuclear factor kappa B kinase subunit beta in Human [GtoPdb: 2039] [UniProtKB: O14920]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
component of inhibitor of nuclear factor kappa B kinase complex in Human [GtoPdb: 1989] [UniProtKB: O15111]
GtoPdb - - 6.19 pKi 650 nM Ki J Med Chem (2017) 60: 7043-7066 [PMID:28737909]
inhibitor of nuclear factor kappa B kinase subunit beta in Human [GtoPdb: 2039] [UniProtKB: O14920]
GtoPdb - - 5.64 pKi 2300 nM Ki J Med Chem (2017) 60: 7043-7066 [PMID:28737909]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.