TP-472 [Ligand Id: 9522] activity data from GtoPdb

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  • bromodomain containing 7 in Human [GtoPdb: 2726] [UniProtKB: Q9NPI1]
Created with Highcharts 10.3.3ValuesChart context menubromodomain containing 7pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2]
Created with Highcharts 10.3.3ValuesChart context menubromodomain containing 9pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 7 in Human [GtoPdb: 2726] [UniProtKB: Q9NPI1]
GtoPdb By isothermal titration calorimetry (ITC). - 6.47 pIC50 340 nM IC50 TP-472 A BRD9/7 Probe. Structural Genomics Consortium.
bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2]
GtoPdb By isothermal titration calorimetry. - 7.48 pIC50 33 nM IC50 TP-472 A BRD9/7 Probe. Structural Genomics Consortium.

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.