miransertib [Ligand Id: 9429] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| AKT serine/threonine kinase 1 in Human [GtoPdb: 1479] [UniProtKB: P31749] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | 5 | nM | IC50 | J Med Chem (2016) 59: 6455-69 [PMID:27305487] |
| GtoPdb | - | - | 8.89 | pIC50 | 1.3 | nM | IC50 | J Med Chem (2022) 65: 14237-14260 [PMID:36197750] |
| AKT serine/threonine kinase 2 in Human [GtoPdb: 1480] [UniProtKB: P31751] | ||||||||
| GtoPdb | - | - | 8.35 | pIC50 | 4.5 | nM | IC50 | J Med Chem (2016) 59: 6455-69 [PMID:27305487] |
| GtoPdb | - | - | 8.85 | pIC50 | 1.4 | nM | IC50 | J Med Chem (2022) 65: 14237-14260 [PMID:36197750] |
| AKT serine/threonine kinase 3 in Human [GtoPdb: 2286] [UniProtKB: Q9Y243] | ||||||||
| GtoPdb | - | - | 7.8 | pIC50 | 16 | nM | IC50 | J Med Chem (2016) 59: 6455-69 [PMID:27305487] |
| GtoPdb | - | - | 8 | pIC50 | 9.9 | nM | IC50 | J Med Chem (2022) 65: 14237-14260 [PMID:36197750] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
