Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CYP3A4 in Human [GtoPdb: 1337] [UniProtKB: P08684] | ||||||||
| GtoPdb | - | - | 6.3 | pIC50 | 500 | nM | IC50 | J Med Chem (2005) 48: 5639-43 [PMID:16134929] |
| Insulin receptor in Human [GtoPdb: 1800] [UniProtKB: P06213] | ||||||||
| GtoPdb | - | - | 7.14 | pIC50 | 73 | nM | IC50 | J Med Chem (2005) 48: 5639-43 [PMID:16134929] |
| Insulin-like growth factor I receptor in Human [GtoPdb: 1801] [UniProtKB: P08069] | ||||||||
| GtoPdb | - | - | 7 | pIC50 | 100 | nM | IC50 | J Med Chem (2005) 48: 5639-43 [PMID:16134929] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.