RA-2 [Ligand Id: 9317] activity data from GtoPdb

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  • KCa2.2 in Mouse [GtoPdb: 382] [UniProtKB: P58390]
Created with Highcharts 10.3.3ValuesChart context menuKCa2.2pKd MousepKi MousepIC50 MousepEC50 Mouse0246810Highcharts.com
  • KCa2.3 in Human [GtoPdb: 383] [UniProtKB: Q9UGI6]
Created with Highcharts 10.3.3ValuesChart context menuKCa2.3pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
KCa2.2 in Mouse [GtoPdb: 382] [UniProtKB: P58390]
GtoPdb - - 7.7 pIC50 20 nM IC50 Mol Pharmacol (2015) 87: 338-48 [PMID:25468883]
KCa2.3 in Human [GtoPdb: 383] [UniProtKB: Q9UGI6]
GtoPdb - - 7.7 pIC50 20 nM IC50 Mol Pharmacol (2015) 87: 338-48 [PMID:25468883]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.