urocortin 1 [Ligand Id: 920] activity data from GtoPdb

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  • CRF1 receptor in Human [GtoPdb: 212] [UniProtKB: P34998]
Created with Highcharts 10.3.3ValuesChart context menuCRF1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • CRF2 receptor in Human [GtoPdb: 213] [UniProtKB: Q13324]
  • CRF2 receptor in Mouse [GtoPdb: 213] [UniProtKB: Q60748]
Created with Highcharts 10.3.3ValuesChart context menuCRF2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 Mouse0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CRF1 receptor in Human [GtoPdb: 212] [UniProtKB: P34998]
GtoPdb - - 9.8 pKd - - - J Pharmacol Exp Ther (2001) 296: 113-20 [PMID:11123370];
Endocrinology (1996) 137: 2167-70 [PMID:8612563];
Nature (1995) 378: 287-92 [PMID:7477349];
J Pharmacol Exp Ther (1999) 288: 729-34 [PMID:9918582];
Proc Natl Acad Sci USA (2001) 98: 7570-5 [PMID:11416224]
CRF2 receptor in Human [GtoPdb: 213] [UniProtKB: Q13324]
GtoPdb - - 9.4 pKd - - - J Pharmacol Exp Ther (2001) 296: 113-20 [PMID:11123370]
CRF2 receptor in Mouse [GtoPdb: 213] [UniProtKB: Q60748]
GtoPdb - - 9.2 pKd - - - Endocrinology (1996) 137: 2167-70 [PMID:8612563];
J Pharmacol Exp Ther (1999) 288: 729-34 [PMID:9918582];
Proc Natl Acad Sci USA (2001) 98: 7570-5 [PMID:11416224]
GtoPdb - - 9.4 pKd - - - J Pharmacol Exp Ther (2001) 296: 113-20 [PMID:11123370];
Endocrinology (1996) 137: 2167-70 [PMID:8612563];
Nature (1995) 378: 287-92 [PMID:7477349];
J Pharmacol Exp Ther (1999) 288: 729-34 [PMID:9918582];
Proc Natl Acad Sci USA (2001) 98: 7570-5 [PMID:11416224]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.